Compound | AgDOP2 | AaDOP2 | CqDOP2 | Fold selectivity to AgDOP2 | |
---|---|---|---|---|---|
AaDOP2 | CqDOP2 | ||||
Amitriptyline | 0.23 ± 0.02 | 0.05 ± 0.003 | 0.08 ± 0.007 | 4.4 | 3.0 |
Amperozide | 18.8 ± 11 | 5.1 ± 1 | 2.6 ± 0.6 | 3.7 | 7.2 |
Asenapine | 0.0007 ± 0.00008 | 0.003 ± 0.0005 | 0.02 ± 0.004 | 0.3 | 0.05 |
Butaclamol | 1.2 ± 0.4 | 1.0 ± 0.2 | 2.8 ± 0.9 | 1.2 | 0.4 |
Chlorprothixene | 0.4 ± 0.007 | 0.04 ± 0.01 | 0.01 ± 0.002 | 0.9 | 3.2 |
Methiothepin | 0.14 ± 0.008 | 0.003 ± 0.001 | 0.01 ± 0.005 | 4.1 | 1.1 |
SCH23390 | 3.6 ± 0.8 | 4.7 ± 0.8 | 8.3 ± 1 | 0.8 | 0.4 |