From: Two old drugs, NVP-AEW541 and GSK-J4, repurposed against the Toxoplasma gondii RH strain
Compound | Parasite inhibition (%) Mean ± SD | Host viability (%) Mean ± SD |
---|---|---|
Atazanavir | 93.6 ± 2.1 | 90.7 ± 2.8 |
PHA-665752 | 92.3 ± 3.1 | 80.5 ± 1.3 |
NVP-AEW541 | 91.5 ± 2.5 | 80.7 ± 1.2 |
Cyclosporine | 90.8 ± 2.1 | 90.4 ± 1.4 |
GSK-J4 HCl | 90.4 ± 1.4 | 92.2 ± 3.8 |
Pemetrexed disodium | 88.9 ± 3.6 | 84.6 ± 1.5 |
Mocetinostat | 86.5 ± 3.1 | 80.2 ± 3.8 |
AMG-208 | 86.4 ± 5.3 | 82.8 ± 1.8 |
CHR2797 | 85.6 ± 1.8 | 88.8 ± 6.7 |
H 89 2HCl | 83.5 ± 1.8 | 89.4 ± 4.6 |
Blonanserin | 82.1 ± 3.1 | 88.3 ± 5.9 |
Lurasidone HCl | 80.4 ± 1.5 | 86.9 ± 1.7 |
ZM 323881 HCl | 79.9 ± 1.4 | 85.5 ± 5.4 |
Pamidronate disodium | 79.6 ± 1.5 | 80.8 ± 1.4 |
Cyproheptadine HCl | 79.2 ± 3.5 | 90.6 ± 1.2 |
Entinostat | 75.7 ± 2.2 | 81.6 ± 1.5 |
Medetomidine HCl | 70.8 ± 1.5 | 90.5 ± 4.4 |
Lafutidine | 70.6 ± 2.5 | 92.7 ± 5.6 |