Wormbase IDa size (aa) GeneDB IDb size (aa) | Human ortholog (% ID) UniProt ID | Structural druggabilityc | Epigenetic inhibitor/ chemical probed |
---|---|---|---|
Smp_150560a (1164) | LSD1 (36%) O60341 | 0.752 | GSK2879552, GSK-LSD1 [51] Tranylcypromine [52] |
Smp_160810a (916) | LSD2 (28%) Q8NB78 | 0.589 | – |
Smp_162940a (1105) | LSD2 (27%) Q8NB78 | 0.543 | – |
Smp_161400a (2575) | KDM3B (46%) Q7LBC6 | 0.766 | JDI‐4 [53] |
Smp_132170a (984) | KDM4C (53%) Q9H3R0 | 0.718 | 4-hydroxypyrazole [54] |
Smp_019170a (1639) | KDM5D (41%) Q9BY66 | 0.891 | – |
Smp_156290a (2612) | KDM5B (47%) Q9UGL1 | 0.848 | KDOAM-25 [55] |
Smp_034000a (1393) | KDM6A (52%) O15550 | 0.921 | GSK-J4 [26] |
Smp_315890a (483) Smp_127230b, e | KDM7A (39%) Q6ZMT4 | 0.84e | Daminozide (N-(dimethylamino) succinamic acid [56] |
Smp_213920a (401) Smp_147870b, e | JMJD4 (40%) Q9H9V9 | 0.801e | – |
Smp_316180a (782) | JMJD6 (61%) Q6NYC1 | 0.857 | – |
Smp_342360a (353) Smp_128500b, e | JMJD5 (41%) Q8N371 | 0.688e | – |
Smp_241580a (396) Smp_180990b, e | JMJD5 (25%) Q8N371 | 0.854e | – |
Smp_333400a (771) Smp_173670b, e | NO66/RIOX1 (26%) Q9H6W3 | 0.764e | – |